longevityfirst-generation GH secretagogue

GHRP-6

GHRP-6 is a synthetic hexapeptide (His-D-Trp-Ala-Trp-D-Phe-Lys-NH2) and the compound that opened the entire growth hormone secretagogue field. It came out of Cyril Bowers' work in the early 1980s on opioid-derived peptides that released growth hormone without acting through GHRH. Every later secretagogue, including GHRP-2, hexarelin, ipamorelin, and the orally active MK-677, descends from this molecule and is usually benchmarked against it.

class
GHRP (hexapeptide secretagogue)
half-life
~15–20 minutes
route
subcutaneous
cadence
2–3x daily, fasted
typical dose
100–300 mcg per injection
cycle
12–16 weeks, then 4-week break
storage
refrigerated · 28-day max (reconstituted)
Dose calculatorlive
U-100
Concentration
2.00mg/mL
Injection vol.
0.050mL
Syringe cap.
100units
Draw to5.0units
0204060801005.0 units
Dosing guide

GHRP-6 Reconstitution & Dosage Protocol

weekly dose · reduces side effects
PhaseWindowWeekly doseDraw (U-100, 2.5mL BAC)Note
IntroductionWeeks 1–20.10 mg5 units· 0.05 mL100 mcg once daily, fasted, to gauge the hunger and facial flush response
StandardWeeks 3–120.10 mg5 units· 0.05 mL100 mcg 2–3x daily (morning fasted, post-training, pre-sleep); stack with a GHRH analog
High outputWeeks 4–120.30 mg15 units· 0.15 mLOptional 300 mcg ceiling during a bulk; hunger becomes the limiting factor before GH does
MaintenanceWeeks 13–160.10 mg5 units· 0.05 mLTaper to 100 mcg once daily before a 4-week washout
How it works

What is GHRP-6?

GHRP-6 is a synthetic hexapeptide (His-D-Trp-Ala-Trp-D-Phe-Lys-NH2) and the compound that opened the entire growth hormone secretagogue field. It came out of Cyril Bowers' work in the early 1980s on opioid-derived peptides that released growth hormone without acting through GHRH. Every later secretagogue, including GHRP-2, hexarelin, ipamorelin, and the orally active MK-677, descends from this molecule and is usually benchmarked against it.

GHRP-6 binds the growth hormone secretagogue receptor (GHS-R1a) in the pituitary and hypothalamus, the receptor whose natural ligand is ghrelin. Receptor activation does two things at once: it directly signals somatotroph cells to release stored growth hormone, and it suppresses somatostatin, the hypothalamic brake on GH output. That dual action is why a GHRP produces a much larger pulse than a GHRH analog used alone.

GHRP-6 does not work in isolation from the GHRH system. A 1998 JCEM study showed that blocking endogenous GHRH sharply reduced the GH response to GHRP-6, meaning the peptide needs intact hypothalamic GHRH signaling to reach its full effect. This is the pharmacological basis for stacking: pairing GHRP-6 with CJC-1295 without DAC or sermorelin produces a synergistic pulse rather than a simply additive one, and it is why the GHRH plus GHRP-6 combination became a standard clinical test for growth hormone deficiency.

The defining practical trait of GHRP-6 is hunger. Of all the GHRPs it produces the most pronounced appetite stimulation, often arriving 20–30 minutes after injection and strong enough to be disruptive for anyone in a caloric deficit. Rodent work showed that centrally administered GHRP-6 drives eating even when plasma GH does not change, confirming that the orexigenic effect is a separate central action and not a downstream consequence of the GH pulse. For a cutting phase, ipamorelin is the correct substitute.

GHRP-6 also raises cortisol and prolactin more than ipamorelin does, though less dramatically than hexarelin at equivalent doses. At 100 mcg per injection the spillover is usually minor. Above roughly 300 mcg the GH response flattens while the cortisol and prolactin curves keep climbing, so raising the dose past that point mostly buys side effects. Transient facial flushing and warmth in the first few minutes after injection are common and harmless.

Common questions

GHRP-6 Frequently Asked Questions

Most protocols use 100 mcg per injection, 2 to 3 times daily, which is close to the saturating dose for GH release in adults (roughly 1 mcg per kg of bodyweight). Some users run up to 300 mcg per injection during a bulking phase. Beyond 300 mcg the GH response plateaus while cortisol, prolactin, and appetite keep increasing, so there is little reason to go higher.
Sources

Research & References

Growth hormone (GH)-releasing peptide-6 requires endogenous hypothalamic GH-releasing hormone for maximal GH stimulationPubMed · J Clin Endocrinol Metab 1998Pharmacokinetic study of growth hormone-releasing peptide 6 (GHRP-6) in nine male healthy volunteersPubMed · Eur J Pharm Sci 2013Effects of a prolonged growth hormone (GH)-releasing peptide infusion on pulsatile GH secretion in normal menPubMed · J Clin Endocrinol Metab 1993Intracerebroventricular growth-hormone-releasing peptide-6 stimulates eating without affecting plasma growth hormone responses in ratsPubMed · Life Sci 1995The GHRH/GHRP-6 test for the diagnosis of GH deficiency in elderly or severely obese menPubMed · Eur J Endocrinol 2005
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